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Your Complete Herbal Supplement Super Store!
DescriptionESTROGENEX - A NATURAL AROMATASE INHIBITOR AND ESTROGEN BLOCKER
ESTROGENEX - is a nutritional supplement, available without a prescription, designed to
normalize all hormone levels, yielding a wide spectrum of health and anti-aging benefits.
ESTROGENEX - is a multi-pathway formulation that minimizes or eliminates the undesirable
effects associated with an estrogen dominant environment.
ESTROGENEX - maintains the correct testosterone to estrogen ratios that yield the benefits
associated with normal estrogen levels.
ESTROGENEX - acts as an irreversible anti-aromatase agent and is thus a powerful elevator of
total testosterone and maximum liberator of free testosterone.
ESTROGENEX - may also play a role in long-term selective estrogen blocking and/or inhibition of
selective estrogen signaling.
ESTROGENEX - may contribute to notable improvements in muscular growth and fat loss, in
addition to its wide array of health and anti-aging benefits.
ESTROGENEX - is designed for: Normalization of all hormone levels, with specific tendencies
toward testosterone dominance, in all aging males.
Prevention and reversal of Gynecomastia.
Adjunctive supplementation for men undergoing hormone replacement therapy to ensure that
raising testosterone levels will not yield an undesirable increase in estrogen levels.
A natural, more effective alternative for traditional testosterone hormone replacement
Bodybuilders and athletes during and immediately after periods of anabolic steroid use for the
purpose of stimulating endogenous testosterone production.
Testosterone: Free-Testosterone and Plasma Protein-Bound Testosterone
Testosterone exists in the blood in either an active (free) or unbound state (+-2%) or inactive
state bound to one of two proteins: sex-hormone-binding-globulin (SHBG) (+-45%) or albumin
(+-53%). Only when testosterone is in its free state can it directly interact with cellular
receptors and exert its activity. SHBG preferentially binds to testosterone over estrogen.
Higher levels of SHBG in women help to maintain higher estrogen to testosterone ratios.
Increased estrogen leads to an increase in SHBG. Thus, lowering the level of SHBG allows for an
increased level of free testosterone. Obviously, if testosterone finds it more difficult to
locate available plasma proteins in the presence of the additional compound, more will be left
in an unbound state.
The amount of free testosterone can be altered (increased) by the use of aromatase inhibitors
(the less testosterone that is synthesized [aromatized] into estrogen, the more total
testosterone) or inhibitors of the plasma proteins that bind into testosterone. Manipulating
the tendency of a testosterone to exist in an unbound state is an effective way to alter the
overall activity and potency of one?s overall testosterone levels. Higher levels of
testosterone produce an enhanced anti-glucocorticoid effect, which yields an anti-catabolic, or
more precisely, anti-proteoolytic, effect on muscle cells. This indirect anabolic effect is the
result of testosterone?s high affinity for binding with glucocorticoid receptors, thus blocking
the normal messenger pathway that triggers protein release from muscle tissue. More free
testosterone also likely results in higher concentrations of IGF-1 and IGF-1 receptor sites in
skeletal muscle tissue. Correspondingly, lower testosterone also likely yields less IGF-1
production and a corresponding decrease in IGF-1 receptor sites. Lower free testosterone also
likely means a weaker immune system.
The Synthesis (Aromatization) of Testosterone to Estrogen in Males and the Significance of
Maintaining Correct Testosterone to Estrogen Ratios.
Although testosterone is considered to be a male hormone and estrogen a female hormone, both
hormones exist in both males and females and serve important functions for both. Estrogen is a
term that really represents a collection of female hormones, with esterone predominating. Since
esterone is the estrogen that is normally in the highest concentration, it is an excellent
marker for basic estrogen levels for that reason. At least three estrogens have multiple and
overlapping functions. Men obtain their estrogen through the action of the aromatase, which
synthesizes (aromatizes) testosterone into estrogen. However, when concentrations of estrogen
become too high and/or the normal ratio of testosterone to estrogen decreases, the potential
for the development of undesirable conditions arises. This includes the development of the
female breast tissue (gynecomastia), increased body fat and water retention. Also, research
suggests that DHT and prostate tissue growth have a direct connection to above normal estrogen
elevations and reduced testosterone levels.
The ESTROGENEX - Mechanism of Action
The ESTROGENEX - proprietary formula was developed by combining naturally occurring aromatase
inhibitors and inhibitors of the action of SHBG. The primary active ingredients in ESTROGENEX
are Coumesterol and Chrysin. ESTROGENEX does not exert its action through any direct hormonal
or prohormonal activity (androgenic or estrogenic).
Before ESTROGENEX , little success had been achieved using chrysin as an effective aromatase
inhibitor because chrysin is poorly absorbed in the bloodstream. However, in addition to their
own specific aromatase inhibiting and estrogen blocking actions, the proprietary blend of other
ingredients work in synergy with chrysin to maintain a stable estrogen environment. We also
incorporated our proprietary delivery system called EXTEND-RX? to avoid competing with other
hormones such as testosterone in the Aromatase Cytochrome P450.
It is believed that ESTROGENEX exerts its effects through several mechanisms of action, which
can be classified into two groups: 1. as an inhibitor of the aromatase enzyme responsible for
the conversion of testosterone to estrogen and an inhibitor of the action of SHBG, and 2. as a
blocker of selective anabolic estrogen receptors and/or inhibitor of selective estrogen
Substances that are aromatase inhibitors block the action of the enzyme aromatase that converts
testosterone to estrogen. Substances that act as an anti-estrogen are those that block the
estrogen receptor. Thus, even though there is estrogen circulating in the blood, the estrogen
cannot exert its effects because it is blocked from attaching to its estrogen receptor. The
dietary supplement ESTROGENEX ? is a multi-pathway agent that exerts its influence by blocking
various stages in the aromatase process and by inhibiting SHBG's action; an activity not
clearly addressed by any of the aromatase inhibiting or anti-estrogen products. Further, it
appears that use of ESTROGENEX may result in long-term blocking of selective anabolic estrogen
receptors and/or inhibition of selective estrogen signaling (these anabolic estrogens are those
demonstrating the undesirable effects associated with breast cancer and gynecomastia). This
activity has not been addressed by any known dietary supplements or pharmacological agents.
ESTROGENEX as an Elevator of Total Testosterone and Liberator of Free Testosterone
As a powerful aromatase inhibitor, ESTROGENEX also possesses notable testosterone stimulating
properties. The aromatase inhibiting action reduces the signal that estrogen sends to the brain
to suppress endogenous testosterone production (estrogen is a main feedback signal to control
the release of testosterone, thus increasing the testicular output of testosterone). ESTROGENEX
thus assists in resetting the body's level of its own natural testosterone production by
regulating the activity of the hypothalamic-pituitary-testicular axis (HPTA), which constantly
adjusts the body's production of testosterone to maintain target blood levels. Continued use of
ESTROGENEX results in not only a significant reduction in the production of estrogen, but also
a corresponding substantial increase in endogenous testosterone.
Only ESTROGENEX addresses all possible channels to estrogen maintenance and free testosterone
elevation, which means optimal hormonal levels for muscle building, fat loss and anti-aging
|Super Lignan, Herbal Estrogen Supplement - Nature's Way, 60 VcapsEFAGold Super Lignan is an ideal herbal estrogen supplement for supporting breast health during the menopausal phases of life helping alleviate breast tenderness and pain associated with the menstrual cycle.|
|Progestacare + Progesterone Cream Pump, For Women, 4 ozProgestaCare Plus combines ProgestaCare's bio-identical progesterone with the highest quality all natural phytoestrogens.|
|Brevail, 6 Units 30 capsBrevail is all-natural and non-prescription, intended for healthy women concerned with breast health and interested in hormonal harmony.|
|ProgestaCare Cream, For Women, 4 ozProgestaCare Natural Progesterone Cream helps women reduce the severity of PMS symptoms lessen the effects of menopause and counter-balance the effects of estrogen dominance, Infertility, Migraines, Fibrocystic Breast, Skin Care, and Acne.|
|Natural Hormone Replacement For Women Over 45, Jonathan Wright, M.D. & J. MorgenthalerFinally, an alternative to conventional hormone replacement therapy - compelling evidence that natural hormone replacement (NHR) provides all the benefits of conventional HRT but with drastically reduced risks of unwanted side effects and cancer.|
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